OPC 21268

CAS No. 131631-89-5

OPC 21268 ( OPC-21268; OPC21268; OPC 21268 )

Catalog No. M17244 CAS No. 131631-89-5

OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 47 In Stock
5MG 72 In Stock
10MG 97 In Stock
25MG 164 In Stock
50MG 230 In Stock
100MG 398 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    OPC 21268
  • Note
    Research use only, not for human use.
  • Brief Description
    OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
  • Description
    OPC-21268 is a vasopressin 1 receptor antagonist potentially for the treatment of heart failure and hypertension.
  • Synonyms
    OPC-21268; OPC21268; OPC 21268
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    DNA/RNA Synthesis
  • Recptor
    Vasopressin receptor 1
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    131631-89-5
  • Formula Weight
    449.55
  • Molecular Formula
    C26H31N3O4
  • Purity
    98%
  • Solubility
    DMSO : 50 mg/mL. 111.22 mM;
  • SMILES
    CC(=O)NCCCOC1=CC=C(C=C1)C(=O)N2CCC(CC2)N3C(=O)CCC4=CC=CC=C43
  • Chemical Name
    N-(3-(4-(4-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)piperidine-1-carbonyl)phenoxy)propyl)acetamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Yamamura Y,etal.PC-21268, an orally effective, nonpeptide vasopressin V1 receptor antagonist.Science. 1991 Apr 26;252(5005):572-4.
molnova catalog
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